Assay ID | Title | Year | Journal | Article |
AID145714 | Inhibition of [3H]nisoxetine binding to norepinephrine (NE) transporter | 1994 | Journal of medicinal chemistry, Apr-15, Volume: 37, Issue:8
| Secondary amine analogues of 3 beta-(4'-substituted phenyl)tropane-2 beta-carboxylic acid esters and N-norcocaine exhibit enhanced affinity for serotonin and norepinephrine transporters. |
AID203943 | Binding affinity of [3H]citalopram for serotonin transporter in monkey | 1994 | Journal of medicinal chemistry, Jun-24, Volume: 37, Issue:13
| The discovery of an unusually selective and novel cocaine analog: difluoropine. Synthesis and inhibition of binding at cocaine recognition sites. |
AID232749 | Selectivity index as ratio of IC50 for 5-HT and DA transporters | 1994 | Journal of medicinal chemistry, Jun-24, Volume: 37, Issue:13
| The discovery of an unusually selective and novel cocaine analog: difluoropine. Synthesis and inhibition of binding at cocaine recognition sites. |
AID65033 | Concentration required to inhibit 50% of radioligand binding ([3H]WIN-35428) to the dopamine (DA) transporter in rat | 1994 | Journal of medicinal chemistry, Sep-02, Volume: 37, Issue:18
| Synthesis, ligand binding, and QSAR (CoMFA and classical) study of 3 beta-(3'-substituted phenyl)-, 3 beta-(4'-substituted phenyl)-, and 3 beta-(3',4'-disubstituted phenyl)tropane-2 beta-carboxylic acid methyl esters. |
AID204374 | Inhibition of [3H]paroxetine binding at serotonin transporter was determined | 2003 | Journal of medicinal chemistry, May-08, Volume: 46, Issue:10
| 2002 Medicinal Chemistry Division Award address: monoamine transporters and opioid receptors. Targets for addiction therapy. |
AID64206 | Displacement of [3H]WIN-35428 from monkey dopamine transporter | 1994 | Journal of medicinal chemistry, Jun-24, Volume: 37, Issue:13
| The discovery of an unusually selective and novel cocaine analog: difluoropine. Synthesis and inhibition of binding at cocaine recognition sites. |
AID64343 | Compounds binding ability to dopamine transporter was evaluated by displacing [3H]beta-CFT in baboon brain | 1993 | Journal of medicinal chemistry, Jun-25, Volume: 36, Issue:13
| Enantioselectivity of cocaine recognition sites: binding of (1S)- and (1R)-2 beta-carbomethoxy-3 beta-(4-iodophenyl)tropane (beta-CIT) to monoamine transporters. |
AID227870 | Tested for its ability to displace [125I]- (1R)-beta-CIT with rat striatal membranes | 1993 | Journal of medicinal chemistry, Jun-25, Volume: 36, Issue:13
| Enantioselectivity of cocaine recognition sites: binding of (1S)- and (1R)-2 beta-carbomethoxy-3 beta-(4-iodophenyl)tropane (beta-CIT) to monoamine transporters. |
AID147749 | Affinity for norepinephrine transporter determined by [3H]nisoxetine displacement. | 2003 | Journal of medicinal chemistry, May-08, Volume: 46, Issue:10
| 2002 Medicinal Chemistry Division Award address: monoamine transporters and opioid receptors. Targets for addiction therapy. |
AID64866 | Inhibition of [3H]WIN-35428 binding at dopamine transporter was determined | 2003 | Journal of medicinal chemistry, May-08, Volume: 46, Issue:10
| 2002 Medicinal Chemistry Division Award address: monoamine transporters and opioid receptors. Targets for addiction therapy. |
AID204376 | Inhibition of [3H]paroxetine binding to 5-hydroxytryptamine (5-HT) transporter | 1994 | Journal of medicinal chemistry, Apr-15, Volume: 37, Issue:8
| Secondary amine analogues of 3 beta-(4'-substituted phenyl)tropane-2 beta-carboxylic acid esters and N-norcocaine exhibit enhanced affinity for serotonin and norepinephrine transporters. |
AID65021 | Potency for the inhibition of [3H]WIN-35428 binding to the dopamine transporter | 1992 | Journal of medicinal chemistry, Mar-20, Volume: 35, Issue:6
| Cocaine receptor: biochemical characterization and structure-activity relationships of cocaine analogues at the dopamine transporter. |
AID220018 | Tested for its ability to displace [125I]- (1R)-beta-CIT with rat cortical membranes | 1993 | Journal of medicinal chemistry, Jun-25, Volume: 36, Issue:13
| Enantioselectivity of cocaine recognition sites: binding of (1S)- and (1R)-2 beta-carbomethoxy-3 beta-(4-iodophenyl)tropane (beta-CIT) to monoamine transporters. |
AID64872 | Inhibition of [3H]WIN-35428 binding to dopamine (DA) transporter | 1994 | Journal of medicinal chemistry, Apr-15, Volume: 37, Issue:8
| Secondary amine analogues of 3 beta-(4'-substituted phenyl)tropane-2 beta-carboxylic acid esters and N-norcocaine exhibit enhanced affinity for serotonin and norepinephrine transporters. |
AID229546 | Relative affinity for norepinephrine and dopamine transporters | 1994 | Journal of medicinal chemistry, Apr-15, Volume: 37, Issue:8
| Secondary amine analogues of 3 beta-(4'-substituted phenyl)tropane-2 beta-carboxylic acid esters and N-norcocaine exhibit enhanced affinity for serotonin and norepinephrine transporters. |
AID204852 | Inhibition of [3H]paroxetine binding at serotonin transporter was determined | 2003 | Journal of medicinal chemistry, May-08, Volume: 46, Issue:10
| 2002 Medicinal Chemistry Division Award address: monoamine transporters and opioid receptors. Targets for addiction therapy. |
AID229540 | Relative affinity for serotonin and dopamine transporters | 1994 | Journal of medicinal chemistry, Apr-15, Volume: 37, Issue:8
| Secondary amine analogues of 3 beta-(4'-substituted phenyl)tropane-2 beta-carboxylic acid esters and N-norcocaine exhibit enhanced affinity for serotonin and norepinephrine transporters. |
AID64845 | Affinity against cocaine binding site of dopamine transporter in rat striatum using [3H]2b as radioligand. | 1991 | Journal of medicinal chemistry, Sep, Volume: 34, Issue:9
| Synthesis, ligand binding, QSAR, and CoMFA study of 3 beta-(p-substituted phenyl)tropane-2 beta-carboxylic acid methyl esters. |
AID204062 | Compounds binding ability to serotonin transporter was evaluated by displacing [3H]paroxetine in baboon brain | 1993 | Journal of medicinal chemistry, Jun-25, Volume: 36, Issue:13
| Enantioselectivity of cocaine recognition sites: binding of (1S)- and (1R)-2 beta-carbomethoxy-3 beta-(4-iodophenyl)tropane (beta-CIT) to monoamine transporters. |
AID147737 | Inhibition of [3H]nisoxetine binding at norepinephrine transporter | 2003 | Journal of medicinal chemistry, May-08, Volume: 46, Issue:10
| 2002 Medicinal Chemistry Division Award address: monoamine transporters and opioid receptors. Targets for addiction therapy. |
[information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |